顔写真

PHOTO

Sako Makoto
佐古　真
Sako Makoto
佐古　真
Institutional repository
Graduate School of Pharmaceutical Sciences　Advanced Pharmaco-science, Assistant Professor
Institutional repository

Research History 2

  1. 2020/05 - Present
    Osaka University　Graduate School of Pharmaceutical Sciences

  2. 2017/04 - 2020/05
    Osaka University　The Institute of Scientific and Industrial Research

Education 4

  1. Osaka University　Graduate School of Science　Department of Chemistry

    2014/04 - 2017/03

  2. Osaka University　Graduate School of Science　Department of Chemistry

    2012/04 - 2014/03

  3. Nara National College of Technology　Faculty of Advanced Engineering Adbanced Chemical Engineerig Course

    2010/04 - 2012/03

  4. Nara National College of Technology　Department of Chemical Engineering

    2005/04 - 2010/03

Committee Memberships 4

  1. 日本薬学会第146年会 一般シンポジウム「有機合成化学の若い力」 世話人（代表）

    2025/04 - Present

  2. NISTEP専門調査員

    2020/04 - Present

  3. 日本薬学会第145年会 一般シンポジウム「有機合成化学の若い力」 世話人

    2024/04 - 2025/03

  4. 第7回アライアンス若手研究交流会 実行委員

    2019/05 - 2019/11

Professional Memberships 5

  1. 一般社団法人 近畿化学協会

  2. ヨウ素学会

  3. 公益社団法人 日本薬学会

  4. 公益社団法人 有機合成化学協会

  5. 公益社団法人 日本化学会

Research Areas 2

  1. Life sciences / Pharmaceuticals - chemistry and drug development /

  2. Nanotechnology/Materials / Synthetic organic chemistry /

Awards 7

  1. 公益財団法人 UBE学術振興財団 第65回学術奨励賞

    2025/04

  2. 令和６年度大阪大学賞（若手教員部門）

    2024/11

  3. 有機合成化学協会 2022年 三菱ガス化学 研究企画賞

    2022/12

  4. The Fourth International Symposium on C–H Activation (ISCHA4) Poster Prize (Asian J. Org. Chem.)

    2018/09

  5. 第6回JACI/GSCシンポジウム GSCポスター賞

    2017/07

  6. Molecular Chirality Asia 2016 Best Poster Prize

    2016/04

  7. 奈良工業高等専門学校専攻科論文発表賞

    2012/03

Papers 48

  1. Multitasking rhodium-catalyzed remote C(sp3)–H functionalization reactions of acyclic dienes to yield benzene-fused heterocycles

    Yuta Sato, Momoko Nagafuchi, Masaharu Takatsuki, Tsuyoshi Matsuzaki, Takeyuki Suzuki, Makoto Sako, Mitsuhiro Arisawa

    Green Chemistry　2024/11/08　Research paper (scientific journal)

    Publisher: Royal Society of Chemistry (RSC)

  2. Brønsted acid-catalyzed synthesis of spirocyclobutanes via heteroannulation of vinyloxyphenylbicyclobutanes with water

    Masaharu Takatsuki, Hiroshi Aoyama, Mitsuhiro Arisawa, Makoto Sako

    Organic & Biomolecular Chemistry　2024/05　Research paper (scientific journal)

    Publisher: Royal Society of Chemistry (RSC)

  3. Axially Chiral Borinic Acid Catalysts: Design, Synthesis, and Application in Alkylative Desymmetrization of 1,2-Diols

    Yuta Chikashige, Tsunayoshi Takehara, Tsuyoshi Matsuzaki, Takeyuki Suzuki, Kenichi Murai, Mitsuhiro Arisawa, Makoto Sako

    The Journal of Organic Chemistry　2023/09/16　Research paper (scientific journal)

    Publisher: American Chemical Society (ACS)

  4. Heteroannulation of bicyclobutane derivatives via Au-catalyzed hydration to enol ethers and intramolecular cyclization giving spirocyclobutanes

    Masaharu Takatsuki, Hiroshi Aoyama, Kenichi Murai, Mitsuhiro Arisawa, Makoto Sako

    Chemical Communications　Vol. 59　No. 48　p. 7467-7470　2023/05　Research paper (scientific journal)

    Publisher: Royal Society of Chemistry (RSC)

  5. Electrochemical Synthesis of Hetero[7]helicenes Containing Pyrrole and Furan Rings via an Oxidative Heterocoupling and Dehydrative Cyclization Sequence

    Mohamed S.H. Salem, Md Imrul Khalid, Makoto Sako, Keigo Higashida, Charlie Lacroix, Masaru Kondo, Ryo Takishima, Taisei Taniguchi, Masahiro Miura, Giang Vo-Thanh, Hiroaki Sasai, Shinobu Takizawa

    Advanced Synthesis and Catalysis　Vol. 365　No. 3　p. 373-380　2023/02/07　Research paper (scientific journal)

  6. Electrochemical synthesis of heterodehydro[7]helicenes

    Md. Imrul Khalid, Mohamed S. H. Salem, Makoto Sako, Masaru Kondo, Hiroaki Sasai, Shinobu Takizawa

    Communications Chemistry　Vol. 5　No. 1　2022/12/03　Research paper (scientific journal)

    Publisher: Springer Science and Business Media LLC

  7. Metal-free C(aryl)–P bond cleavage: experimental and computational studies of the Michael addition/aryl migration of triarylphosphines to alkynyl esters

    Makoto Sako, Kyohei Kanomata, Mohamed S. H. Salem, Tomohiro Furukawa, Hiroaki Sasai, Shinobu Takizawa

    Organic Chemistry Frontiers　Vol. 9　No. 8　p. 2187-2192　2022/03　Research paper (scientific journal)

    Publisher: Royal Society of Chemistry (RSC)

  8. Chemo- and enantioselective hetero-coupling of hydroxycarbazoles catalyzed by a chiral vanadium(v) complex

    Makoto Sako, Keigo Higashida, Ganesh Tatya Kamble, Kevin Kaut, Ankit Kumar, Yuka Hirose, Da-Yang Zhou, Takeyuki Suzuki, Magnus Rueping, Tomohiro Maegawa, Shinobu Takizawa, Hiroaki Sasai

    Organic Chemistry Frontiers　Vol. 8　No. 17　p. 4878-4885　2021/06/23　Research paper (scientific journal)

    Publisher: Royal Society of Chemistry ({RSC})

  9. Recent Advances in Metal-Nanoparticle-Catalyzed Coupling Reactions Assisted by Microwave Irradiation

    Makoto Sako, Mitsuhiro Arisawa

    Synthesis　Vol. 53　No. 19　p. 3513-3521　2021/05/10　Research paper (scientific journal)

    Publisher: Georg Thieme Verlag {KG}

  10. Chiral vanadium complex-catalyzed oxidative coupling of arenols

    Makoto Sako, Shinobu Takizawa, Hiroaki Sasai

    Tetrahedron　Vol. 76　No. 47　p. 131645-131645　2020/10/07　Research paper (scientific journal)

    Publisher: Elsevier {BV}

  11. Catalytic and Enantioselective oxa-Piancatelli Reaction Using Chiral Vanadium Complex

    Makoto Sako

    Chemical Communications　2020/07/23　Research paper (scientific journal)

    Publisher: Royal Society of Chemistry (RSC)

  12. C–H Triflation of BINOL Derivatives Using DIH and TfOH

    Nakazawa, H, Sako, M, Masui, Y, Kurosaki, R, Yamamoto, S, Kamei, T, Shimada, T

    Organic Letters　2019/08/06　Research paper (scientific journal)

  13. Chiral Dinuclear Vanadium Complex-Mediated Oxidative Coupling of Resorcinols

    Makoto Sako, Takanori Aoki, Nadine Zumbrägel, Lukas Schober, Harald Gröger, Shinobu Takizawa, Hiroaki Sasai

    The Journal of Organic Chemistry　Vol. 84　No. 3　p. 1580-1587　2018/12/06　Research paper (scientific journal)

    Publisher: American Chemical Society ({ACS})

  14. Chiral Vanadium Complex-catalyzed Enantioselective Oxidative Coupling Reactions

    Makoto Sako, Shinobu Takizawa, Hiroaki Sasai

    Journal of Synthetic Organic Chemistry, Japan　Vol. 76　No. 9　p. 874-884　2018/09/01　Research paper (scientific journal)

    Publisher: The Society of Synthetic Organic Chemistry, Japan

  15. Vanadium-Catalyzed Dehydrogenation of N-Heterocycles in Water

    Zumbrägel, N., Sako, M., Takizawa, S., Sasai, H., Gröger, H.

    Organic Letters　Vol. 20　No. 16　p. 4723-4727　2018/08/17　Research paper (scientific journal)

    Publisher: American Chemical Society ({ACS})

  16. Enantio- and Diastereoselective Betti/aza-Michael Sequence: Single Operated Preparation of Chiral 1,3-Disubstituted Isoindolines

    Shinobu Takizawa, Makoto Sako, Mohamed Ahmed Abozeid, Kenta Kishi, H. D. P. Wathsala, Shuichi Hirata, Kenichi Murai, Hiromichi Fujioka, Hiroaki Sasai

    Organic Letters　Vol. 19　No. 19　p. 5426-5429　2017/09/28　Research paper (scientific journal)

  17. Short Syntheses of 4-Deoxycarbazomycin B, Sorazolon E, and (+)-Sorazolon E2

    Makoto Sako, Kazuya Ichinose, Shinobu Takizawa, Hiroaki Sasai

    Chemistry - An Asian Journal　Vol. 12　No. 12　p. 1305-1308　2017/05　Research paper (scientific journal)

  18. Efficient Enantioselective Synthesis of Oxahelicenes Using Redox/Acid Cooperative Catalysts

    Makoto Sako, Yoshiki Takeuchi, Tetsuya Tsujihara, Junpei Kodera, Tomikazu Kawano, Shinobu Takizawa, Hiroaki Sasai

    Journal of the American Chemical Society　Vol. 138　No. 36　p. 11481-11484　2016/08　Research paper (scientific journal)

  19. Total Synthesis of (±)-Minimiflorin and Its Na+/K+-ATPase and H+/K+-ATPase Inhibitory Activities

    Wataru Yamawaki, Kuniaki Suzuki, Yuri Hase, Hiroshi Aoyama, Atsushi Nakayama, Makoto Sako, Mitsuhiro Arisawa

    Journal of Natural Products　2025/06/29　Research paper (scientific journal)

    Publisher: American Chemical Society (ACS)

  20. Synthesis of Dibenzoxasilepine Using Ring Expansion Reaction of a Pentacoordinate Silicon Intermediate

    Keigo WATANABE, Mutsuki Sato, Tsunayoshi Takehara, Kaori ASANO, Tsuyoshi Matsuzaki, Takeyuki Suzuki, Makoto SAKO, Mitsuhiro Arisawa

    Advanced Synthesis & Catalysis　2024/11/26　Research paper (scientific journal)

    Publisher: Wiley

  21. Absorption, Fluorescence, and Two-Photon Excitation Ability of 5-o-Tolyl-11 (or 13)-o-tolylisoindolo[2,1-a]quinolines Prepared by Ring-Closing Metathesis and [2+3] Cycloaddition.

    Yuki Wada, Kwangkyun Jang, Hirokazu Ishii, Yuki Watakabe, Motosuke Tsutsumi, Makoto Sako, Tsunayoshi Takehara, Takeyuki Suzuki, Hirofumi Tsujino, Yasuo Tsutsumi, Tomomi Nemoto, Mitsuhiro Arisawa

    Chemistry, an Asian journal　2024/11/04　Research paper (scientific journal)

  22. Oxidative Rearrangement Approach for the Ring Contraction of N−H Piperidines to Pyrrolidines

    Mirei Takashima, Makoto Miyoshi, Makoto Sako, Mitsuhiro Arisawa, Kenichi Murai

    Advanced Synthesis and Catalysis　Vol. 366　No. 15　p. 3325-3331　2024/08/06　Research paper (scientific journal)

  23. Synthesizing Silyl Arylsulfonyl Hydrazones as Silyldiazomethane Precursors and Their Use in Rhodium‐Catalyzed Reactions

    Shuji Tsuruda, Keigo Saito, Tsuyoshi Matsuzaki, Da‐Yang Zhou, Takeyuki Suzuki, Makoto Sako, Mitsuhiro Arisawa, Kenichi Murai

    Advanced Synthesis & Catalysis　2024/04/17　Research paper (scientific journal)

    Publisher: Wiley

  24. Palladium-Catalyzed Intramolecular Migratory Cycloisomerization of 3-Phenoxy Acrylic Acid Ester <i>via</i> C–O Bond Cleavage and C–O/C–C Bonds Formation for 2,3-Disubstituted Benzofurans Synthesis

    Yuichi Kuboki, Shohei Ohno, Makoto Sako, Kenichi Murai, Mitsuhiro Arisawa

    Chemical and Pharmaceutical Bulletin　Vol. 71　No. 2　p. 93-100　2023/02/01　Research paper (scientific journal)

    Publisher: Pharmaceutical Society of Japan

  25. Total Synthesis of Ansellone G and Phorbadione.

    Mizushi Yanagihara, Kanae Nakahara, Naoki Kishimoto, Towa Abe, Satoshi Miura, Shogo Misumi, Makoto Sako, Mitsuhiro Arisawa, Kenichi Murai

    The Journal of organic chemistry　Vol. 87　No. 24　p. 16913-16917　2022/12/07　Research paper (scientific journal)

  26. Double Ring Expansion Strategy for Fused 3-Benzazepines: Alternative Synthesis of the Dolby-Weinreb Enamine.

    Keigo Saito, Hiroshi Aoyama, Makoto Sako, Mitsuhiro Arisawa, Kenichi Murai

    The Journal of organic chemistry　Vol. 87　No. 24　p. 16947-16951　2022/12/07　Research paper (scientific journal)

  27. Design, Synthesis, and Monoamine Oxidase B Selective Inhibitory Activity of N-Arylated Heliamine Analogues

    Makito Yamada, Yu Hirose, Bangzhong Lin, Megumi Fumimoto, Kazuto Nunomura, Sirimangkalakitti Natchanun, Naoyuki Takahashi, Yuuta Ohki, Makoto Sako, Kenichi Murai, Kazuo Harada, Masayoshi Arai, Sayo Suzuki, Tomonori Nakamura, Junichi Haruta, Mitsuhiro Arisawa

    ACS Medicinal Chemistry Letters　2022/08/22　Research paper (scientific journal)

    Publisher: American Chemical Society (ACS)

  28. Carbon(sp 2 )‐carbon(sp 3 ) Bond‐forming Cross‐coupling Reactions Using Sulfur‐Modified Au‐Supported Nickel Nanoparticle Catalyst

    Ryousuke Ohta, Yasunori Shio, Toshiki Akiyama, Makito Yamada, Shuhei Shimoda, Kazuo Harada, Makoto Sako, Jun‐ya Hasegawa, Mitsuhiro Arisawa

    Asian Journal of Organic Chemistry　2022/07/13　Research paper (scientific journal)

    Publisher: Wiley

  29. Double isomerization/cycloisomerization/aromatization of 1-(allyloxy)-2-(cyclopropylmethyl)benzenes to give 2-ethyl-3-isopropylbenzofurans using a multitasking single rhodium catalyst

    Yuta Sato, Tsuyoshi Matsuzaki, Tsunayoshi Takehara, Makoto Sako, Takeyuki Suzuki, Mitsuhiro Arisawa

    Chemical Communications　2022/01　Research paper (scientific journal)

    Publisher: Royal Society of Chemistry (RSC)

  30. Chemo- and regioselective cross-dehydrogenative coupling reaction of 3-hydroxycarbazoles with arenols catalyzed by a mesoporous silica-supported oxovanadium

    Kengo Kasama, Kyohei Kanomata, Yuya Hinami, Karin Mizuno, Yuta Uetake, Toru Amaya, Makoto Sako, Shinobu Takizawa, Hiroaki Sasai, Shuji Akai

    RSC Advances　Vol. 11　No. 56　p. 35342-35350　2021/11/02　Research paper (scientific journal)

    Publisher: Royal Society of Chemistry ({RSC})

  31. Product selective reaction controlled by the combination of palladium nanoparticles, continuous microwave irradiation, and a co-existing solid; ligand-free Buchwald–Hartwig amination vs. aryne amination

    Makito Yamada, Ryousuke Ohta, Kazuo Harada, Tsunayoshi Takehara, Hitoshi Haneoka, Yosuke Murakami, Takeyuki Suzuki, Yuuta Ohki, Naoyuki Takahashi, Toshiki Akiyama, Natchanun Sirimangkalakitti, Makoto Sako, Kenichi Murai, Masayoshi Arai, Mitsuhiro Arisawa

    Green Chemistry　Vol. 23　No. 20　p. 8131-8137　2021/08/31　Research paper (scientific journal)

  32. Carbon–Carbon Bond Formation between N-Heterocyclic Carbene Ligand on Ruthenium Carbene Catalysts and 1,4-Naphthoquinone via Intramolecular Carbon(sp3)–Hydrogen Bond Activation

    Yuki Wada, Tsunayoshi Takehara, Takeyuki Suzuki, Satoshi Aoki, Takayuki Hibi, Makoto Sako, Hirofumi Tsujino, Yasuo Tsutsumi, Mitsuhiro Arisawa

    Organometallics　Vol. 40　No. 16　p. 2901-2908　2021/08/09　Research paper (scientific journal)

  33. Chiral Vanadium(V)-catalyzed Oxidative Coupling of 4-Hydroxycarbazoles

    Ganesh T. Kamble, Mohamed S. H. Salem, Tsukasa Abe, Hanseok Park, Makoto Sako, Shinobu Takizawa, Hiroaki Sasai

    Chemistry Letters　Vol. 50　No. 10　p. 1755-1757　2021/07/15　Research paper (scientific journal)

    Publisher: The Chemical Society of Japan

  34. Iridium-Catalyzed Isomerization/Cycloisomerization/Aromatization of N-Allyl-N-sulfonyl-o-(λ1-silylethynyl)aniline Derivatives to Give Substituted Indole Derivatives

    Jiawei Qiu, Makoto Sako, Tomoyuki Tanaka, Tsuyoshi Matsuzaki, Tsunayoshi Takehara, Takeyuki Suzuki, Shohei Ohno, Kenichi Murai, Mitsuhiro Arisawa

    Organic Letters　Vol. 23　No. 11　p. 4284-4288　2021/05/25　Research paper (scientific journal)

    Publisher: American Chemical Society ({ACS})

  35. Preparation of Optically Pure Dinuclear Cobalt(III) Complex with Λ-Configuration as a Dianionic Chiral Catalyst

    Mohamed S. H. Salem, Ankit Kumar, Makoto Sako, Tsukasa Abe, Shinobu Takizawa, and Hiroaki Sasai

    HETEROCYCLES　Vol. 103　No. 1　p. 225-225　2020/12/03　Research paper (scientific journal)

    Publisher: The Japan Institute of Heterocyclic Chemistry

  36. Vanadium(V) Complex-Catalyzed One-Pot Synthesis of Phenanthridines via a Pictet-Spengler-Dehydrogenative Aromatization Sequence

    Makoto Sako, Romain Losa, Tomohiro Takiishi, Giang Vo-Thanh, Shinobu Takizawa, Hiroaki Sasai

    Catalysts　Vol. 10　No. 8　p. 860-860　2020/08/02　Research paper (scientific journal)

    Publisher: {MDPI} {AG}

  37. Enantioconvergent Catalytic SN1 Reaction by Stereocontrol over Tertiary Carbocations

    Makoto Sako

    Journal of Synthetic Organic Chemistry, Japan　2020/01/01

  38. Exploration of flow reaction conditions using machine-learning for enantioselective organocatalyzed Rauhut–Currier and [3+2] annulation sequence

    Masaru Kondo, H. D. P. Wathsala, Makoto Sako, Yutaro Hanatani, Kazunori Ishikawa, Satoshi Hara, Takayuki Takaai, Takashi Washio, Shinobu Takizawa, Hiroaki Sasai

    Chemical Communications　2019/12/09　Research paper (scientific journal)

  39. キラルバナジウム触媒によるヘリセン様化合物の簡便合成

    佐古真, 滝澤忍, 笹井宏明

    生産と技術　2019/04

  40. Asymmetric oxidative coupling of hydroxycarbazoles: Facile synthesis of (+)-bi-2-hydroxy-3-methylcarbazole

    Makoto Sako, Akimasa Sugizaki, Shinobu Takizawa

    Bioorganic & Medicinal Chemistry Letters　Vol. 28　No. 16　p. 2751-2753　2018/02　Research paper (scientific journal)

    Publisher: Elsevier {BV}

  41. Chiral organocatalyzed intermolecular Rauhut–Currier reaction of nitroalkenes with ethyl allenoate

    Takizawa, S., Sako, M., Kishi, K., Shigenobu, M., Vo-Thanh, G., Sasai, H.

    Chemical and Pharmaceutical Bulletin　Vol. 65　No. 11　p. 997-999　2017/11　Research paper (scientific journal)

  42. Organocatalyzed [4+2] Annulation of All-Carbon Tetrasubstituted Alkenes with Allenoates: Synthesis of Highly Functionalized 2H- and 4H-Pyran Derivatives.

    Thi-Thuy-Duong Ngo, Kenta Kishi, Makoto Sako, Masashi Shigenobu, Chloée Bournaud, Martial Toffano, Régis Guillot, Jean-Pierre Baltaze, Shinobu Takizawa, Hiroaki Sasai, Giang Vo-Thanh

    ChemistrySelect　Vol. 1　No. 17　p. 5414-5420　2016/10　Research paper (scientific journal)

  43. Asymmetric BrOnsted Acid Catalyzed Substitution of Diaryl Methanols with Thiols and Alcohols for the Synthesis of Chiral Thioethers and Ethers

    Adisak Chatupheeraphat, Hsuan-Hung Liao, Steffen Mader, Makoto Sako, Hiroaki Sasai, Iuliana Atodiresei, Magnus Rueping

    ANGEWANDTE CHEMIE-INTERNATIONAL EDITION　Vol. 55　No. 15　p. 4803-4807　2016/03　Research paper (scientific journal)

  44. An enantioselective organocatalyzed aza-Morita-Baylis-Hillman reaction of isatin-derived ketimines with acrolein

    Yasushi Yoshida, Makoto Sako, Kenta Kishi, Hiroaki Sasai, Susumi Hatakeyama, Shinobu Takizawa

    ORGANIC & BIOMOLECULAR CHEMISTRY　Vol. 13　No. 34　p. 9022-9028　2015/07　Research paper (scientific journal)

  45. Enantioselective and aerobic oxidative coupling of 2-naphthol derivatives using chiral dinuclear vanadium(V) complex in water

    Makoto Sako, Shinobu Takizawa, Yasushi Yoshida, Hiroaki Sasai

    Tetrahedron: Asymmetry　Vol. 26　No. 12-13　p. 613-616　2015/05　Research paper (scientific journal)

  46. Enantioselective construction of C2-symmetric spiro skeleton through intramolecular copper-catalyzed N-arylation

    Kazuhiro Takenaka, Makoto Sako, Shuhei Takatani, Hiroaki Sasai

    Arkivoc　Vol. 2015　No. 2　p. 52-63　2014/11/21　Research paper (scientific journal)

    Publisher: Arkat

  47. Enantioselective oxidative-coupling of polycyclic phenols

    Shinobu Takizawa, Junpei Kodera, Yasushi Yoshida, Makoto Sako, Stefanie Breukers, Dieter Enders, Hiroaki Sasai

    Tetrahedron　Vol. 70　No. 9　p. 1786-1793　2014/03　Research paper (scientific journal)

  48. Scandium triflate-catalyzed 6,6 '-diiodination of 2,2 '-dimethoxy-1,1 '-binaphthyl with 1,3-diiodo-5,5-dimethylhydantoin

    Toshiyuki Kamei, Hiroshi Shibaguchi, Makoto Sako, Kenji Toribatake, Toyoshi Shimada

    TETRAHEDRON LETTERS　Vol. 53　No. 30　p. 3894-3896　2012/07　Research paper (scientific journal)

Misc. 18

  1. アーヘン工科大学での研究と生活（海外研究室レポート）

    佐古真

    Organometallic News　Vol. 3　p. 82-83　2021

  2. 第三級カルボカチオンの立体制御によるエナンチオ収束型触媒的SN1反応（Review de Debut）

    佐古真

    有機合成化学協会誌　Vol. 78　No. 1　p. 60-61　2018

  3. ベンゼンの触媒的非対称化を鍵とするパンクラチスタチン類の不斉全合成

    佐古真

    ファルマシア　Vol. 54　No. 7　2018

  4. ビナフチル化合物のヨウ素化とその利用

    亀井稔之, 佐古真, 嶋田豊司

    SIS Letters　Vol. 14　p. 2-11　2013

  5. Design and Synthesis of Spliceostatin A Derivatives: Structure-Activity-Relationship Study related to Enone moiety of Spliceostatin A

    平林怜, 太田徳子, 露口結子, LI Yue, 吉川祐介, LIN Bangzhong, 文元めぐみ, 春田純一, 佐古真, 村井健一, 二村圭祐, 有澤光弘

    日本化学会春季年会講演予稿集(Web)　Vol. 103rd　2023

  6. 毒性低減化を目指したSpliceostatin A誘導体の設計・合成と機能評価

    平林怜, 吉川祐介, 石橋亜衣里, 佐古真, 村井健一, 金田安史, 二村圭祐, 有澤光弘

    反応と合成の進歩シンポジウム講演要旨集　Vol. 48th　2022

  7. A Chiral Vanadium(V) Complex-Catalyzed Enantioselective Oxidative Coupling of Hydroxycarbazoles

    KAMBLE Ganesh Tatya, SALEM Mohamed S. H., SUGIZAKI Akimasa, PARK Hanseok, SAKO Makoto, TAKIZAWA Shinobu, SASAI Hiroaki

    日本化学会春季年会講演予稿集(Web)　Vol. 102nd　2022

  8. 分子から窒素を引っこ抜け！第二級アミンの分子骨格編集反応の開発（注目の論文）

    佐古真

    化学　Vol. 76　No. 10　p. 66-67　2021

  9. Electrochemical Synthesis of Azaoxa[7]helicenes via Oxidative Hetero-coupling/Dehydrative Cyclization Sequence of Arenols

    SALEM Mohamed S. H., KHALID Md. Imrul, SAKO Makoto, TAKIZAWA Shinobu, SASAI Hiroaki

    日本化学会春季年会講演予稿集(Web)　Vol. 101st　2021

  10. Sequential electrochemical synthesis of cyclic dehydrooxahelicenes

    SALEM Mohamed S. H., KHALID Md. Imrul, SAKO Makoto, KONDO Masaru, TAKIZAWA Shinobu, SASAI Hiroaki

    複素環化学討論会講演要旨集　Vol. 50th　2021

  11. Catalytic Enantioselective Sequential C-C Bond Forming Reaction in Flow System

    WATHSALA H.D.P., KISHI Kenta, CHEN Qingwen, SAKO Makoto, TAKIZAWA Shinobu, SASAI Hiroaki

    日本化学会春季年会講演予稿集(CD-ROM)　Vol. 98th　2018

  12. Vanadium complex catalyzed enantioselective synthesis of oxa[9]helicenes

    Shinobu Takizawa, Makoto Sako, Hiroaki Sasai

    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY　Vol. 251　2016/03　Research paper, summary (international conference)

  13. 5価バナジウム触媒を活用するオキサ[9]ヘリセンのエナンチオ選択的合成

    滝澤忍, 佐古真, 武内芳樹, 辻原哲也, 小寺純平, 河野富一, 笹井宏明

    複素環化学討論会講演要旨集　Vol. 45th　2015

  14. バナジウム触媒を活用するエナンチオ選択的炭素-炭素結合形成反応の開発と応用

    佐古真, 武内芳樹, 滝澤忍, 辻原哲也, 吉田泰志, 小寺純平, 河野富一, 笹井宏明

    有機合成シンポジウム講演要旨集　Vol. 107th　2015

  15. バナジウム触媒を活用するヘテロヘリセン誘導体のエナンチオ選択的合成法の開発

    一之瀬和弥, 佐古真, 武内芳樹, 滝澤忍, 辻原哲也, 小寺純平, 河野富一, 笹井宏明

    反応と合成の進歩シンポジウム講演要旨集　Vol. 41st　2015

  16. 5価のバナジウム触媒を用いるエナンチオ選択的炭素-炭素結合形成反応の開発と応用

    滝澤忍, 辻原哲也, 小寺純平, 秋田三俊, 吉田泰志, 佐古真, 土井貴裕, 畠中稔, 笹井宏明

    日本化学会講演予稿集　Vol. 94th　No. 4　2014

  17. ヘリセン及びヘリセン様化合物の効率的不斉合成法の開発

    滝澤忍, 吉田泰志, 小寺純平, 佐古真, 土井貴裕, 笹井宏明

    シンポジウム「モレキュラー・キラリティー」講演要旨集　Vol. 2014　2014

  18. ヘリセン及びヘリセン様化合物のエナンチオ選択的効率合成法の開発

    滝澤忍, 辻原哲也, 吉田泰志, 小寺純平, 佐古真, 土井貴裕, 笹井宏明

    反応と合成の進歩シンポジウム講演要旨集　Vol. 40th　2014

Publications 1

  1. Chapter 18: Vanadium-catalyzed Enantioselective C–C Bond-forming Reactions

    Makoto Sako, Shinobu Takizawa, Hiroaki Sasai

    Royal Society of Chemistry　2019

Presentations 13

  1. Development of Binaphthyl-type Chiral Borinic Acid Catalysts and Their Application to Catalytic Enantioselective Reaction

    Makoto Sako, Yuta Chikashige, Kazuhiro Higashi, Shuta Mizuse, Tsunayoshi Takehara, Takeyuki Suzuki, Kenichi Murai, Mitsuhiro Arisawa

    2025/05/30

  2. Synthesis of Heterocyclic Compounds Based on Sequential Reactions

    Makoto SAKO

    Vortrag im Rahmen des Organisch-Chemischen IOCB-Kolloquiums (Invited Lecture)　2024/10/09

  3. ヘテロ[ サーキュレンの電解合成と光触媒としての応用

    佐古真, Ahmed S. Gabr, Mohamed S. H. Salem, Md. Imrul Khalid, 滝澤忍

    第1 6 回有機触媒シンポジウム　2023/11/27

  4. スピロシクロブタンを有するヘテロ環合成法の開発：ビシクロブタン誘導体を用いる環形成反応

    佐古 真

    第７回 関西薬学シンポジウム：化学系の若い力　2023/09/16

  5. 機械学習を活用する溶媒効果の定量的説明：極性転換型有機分子触媒反応における検証

    佐古 真, 赤澤 龍之介, 鹿又 喬平, 赤井 周司, 有澤 光弘, 滝澤 忍

    第21回次世代を担う有機化学シンポジウム　2023/05/27

  6. “Au-catalyzed intramolecular cyclization of bicyclobutane derivatives” and “design, synthesis, and evaluation of novel chiral borinic acid catalysts”

    Mini-Symposium on Organic Chemistry　2022/09/21

  7. Chiral Vanadium Complex-mediated oxa-Piancatelli Reaction and Pictet–Spengler Reaction/Aromatization Sequence

    13th International CeBiTec Symposium - Multi-Step Syntheses in Biology & Chemistry, An International Young Investigator Conference -　2019/12/03

  8. キラルバナジウム触媒を用いるフェノール類の酸化的ヘテロカップリング反応

    佐古真, 東田恵伍, 滝澤忍, 笹井宏明

    第66回有機金属化学討論会　2019/09/14

  9. キラルバナジウム錯体の酸触媒能を活用する不斉反応の開発

    佐古真, 瀧石朋大, Lukas Schober, Harald Gröger, 滝澤忍, 笹井宏明

    シンポジウム モレキュラー・キラリティー2019　2019/06/14

  10. Chiral Dinuclear Vanadium Complex-mediated Oxidative Coupling of Monocyclic Phenols

    Sako, M, Aoki, T, Takizawa, S, Sasai, H

    43rd International Conference on Coordination Chemistry (ICCC 2018)　2018/08/03

  11. バナジウム触媒を用いる不斉酸化的カップリング反応の開発と応用

    佐古真, 滝澤忍, 笹井宏明

    第47回複素環化学討論会　2017/10/28

  12. Chiral Vanadium(V) Complex-catalyzed Enantioselective Oxidative Coupling of Phenol Derivatives

    佐古真, 青木孝憲, 滝澤忍, 笹井宏明

    第64回有機金属化学討論会　2017/09/08

  13. バナジウム触媒を活用するエナンチオ選択的炭素－炭素結合形成反応の開発と応用

    佐古真, 武内芳樹, 滝澤忍, 辻原哲也, 吉田泰志, 小寺純平, 河野富一, 笹井宏明

    第107回有機合成シンポジウム　2015/06/10

Industrial Property Rights 2

  1. 新規なデヒドロヘテロヘリセン化合物およびその製造方法

    滝澤 忍, 笹井 宏明, 佐古 真, 近藤 健, カーリド エムディ イムルル

    出願日:2020/11/13

  2. 抗ウイルス作用を有するインドール誘導体

    有澤 光弘, 佐古 真, 上村 健太朗, 田鍬 修平, 松浦 善治, 岡林 環樹

    出願日:2025/03/21

Institutional Repository 3

Content Published in the University of Osaka Institutional Repository (OUKA)

  1. Absorption, Fluorescence, and Two-Photon Excitation Ability of 5-o-Tolyl-11 (or 13)-o-tolylisoindolo[2,1-a]quinolines Prepared by Ring-Closing Metathesis and [2+3] Cycloaddition

    Wada Yuki, Jang Kwangkyun, Ishii Hirokazu, Watakabe Yuki, Tsutsumi Motosuke, Sako Makoto, Takehara Tsunayoshi, Suzuki Takeyuki, Tsujino Hirofumi, Tsutsumi Yasuo, Nemoto Tomomi, Arisawa Mitsuhiro

    Chemistry - An Asian Journal　Vol. 20　No. 2　2025/01/17

  2. Synthesis of Dibenzoxasilepine Using Ring Expansion Reaction of a Pentacoordinate Silicon Intermediate

    Watanabe Keigo, Sato Mutsuki, Takehara Tsunayoshi, Asano Kaori, Matsuzaki Tsuyoshi, Suzuki Takeyuki, Sako Makoto, Arisawa Mitsuhiro

    Advanced Synthesis and Catalysis　2024/12/16

  3. Carbon(sp2)-carbon(sp3) Bond-forming Cross-coupling Reactions Using Sulfur-Modified Au-Supported Nickel Nanoparticle Catalyst

    Ohta Ryousuke, Shio Yasunori, Akiyama Toshiki, Yamada Makito, Shimoda Shuhei, Harada Kazuo, Sako Makoto, Hasegawa Junya, Arisawa Mitsuhiro

    Asian Journal of Organic Chemistry　Vol. 11　No. 9　2022/06/27